


Total Pages: 118
Topics Covered:
Pharmacology Section
• Scientists’ Contributions
• Basic Definitions (Pharmacology, Pharmacodynamics, Pharmacokinetics, Toxicology, etc.)
• Pharmacokinetics (Absorption, Distribution, Metabolism, Excretion)
• Pharmacodynamics & Mechanism of Drug Action
• Drug Interactions, Tolerance & Resistance
• Adverse Drug Reactions (Type A & B, Teratogenicity, Carcinogenicity, etc.)
• Cholinergic System & Drugs (Agonists, Anticholinesterases, Anticholinergics)
• Adrenergic System & Drugs (Sympathomimetics, Antiadrenergics, β-blockers)
• Histamine & Antihistaminics
• 5-HT (Serotonin) & Antagonists
• Drug Therapy of Migraine
• Prostaglandins, Leukotrienes, Platelet Activating Factor
• NSAIDs & Antipyretic-Analgesics
• Antirheumatoid Drugs & DMARDs
• Drugs Used in Gout
• Drugs for Cough & Bronchial Asthma
• Pituitary Hormones (GH, ACTH, Prolactin)
• Thyroid Hormones & Inhibitors
• Insulin & Oral Hypoglycemics
• Corticosteroids
• Androgens & Drugs for Erectile Dysfunction
• Estrogens, Progestins & Contraceptives
• Oxytocin & Uterine Drugs
• Drugs Affecting Calcium Balance (Calcitonin, Vitamin D, Bisphosphonates)
• Skeletal Muscle Relaxants
Medicinal Chemistry Highlights (Integrated SAR Points)
• Structural features of Aspirin & other NSAIDs (COX selectivity, prodrug forms like Sulindac)
• Chemistry & selectivity of β-blockers (1st, 2nd, 3rd generation)
• Salicylates, Propionic acid derivatives, Oxicam & Pyrazolone chemistry notes
• Diuretic features (–SO₂NH₂ group importance, chondroprotective action of Aceclofenac)
• Steroidal vs Non-steroidal estrogen/progestin compounds
• Corticosteroid nucleus & modifications affecting activity
• Insulin analogues & recombinant DNA preparation insights